Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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EPHA7

RBC: EPHA7 · Substrate: pEY · medium confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Ponatinib96.10.53
Cabozantinib92.90.75
Repotrectinib85.80.61
Selpercatinib84.00.64
Tivozanib83.30.67
Crizotinib83.00.58
Fostamatinib82.30.61
Gilteritinib72.20.51
Vandetanib68.00.72
Defactinib66.50.45
Ripretinib56.90.67
Pralsetinib48.60.64
Canertinib48.00.67
Afatinib39.50.71
Dacomitinib39.00.66

Known variants

No variants catalogued.
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