BRSK2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Midostaurin | 94.6 | 0.50 |
| Repotrectinib | 91.5 | 0.61 |
| Brigatinib | 77.8 | 0.51 |
| Axitinib | 76.0 | 0.69 |
| Rabusertib | 56.9 | 0.69 |
| Sunitinib | 43.6 | 0.52 |
| Defactinib | 31.9 | 0.45 |
| Dabrafenib | 23.8 | 0.63 |
| Selpercatinib | 22.3 | 0.64 |
| Abrocitinib | 21.3 | 0.58 |
| Crizotinib | 21.1 | 0.58 |
| Lorlatinib | 20.1 | 0.69 |
| Netarsudil | 17.1 | 0.68 |
| Dacomitinib | 16.7 | 0.66 |
| Paxalisib | 14.4 | 0.61 |
Known variants
No variants catalogued.