Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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EPHA5

RBC: EPHA5 · Substrate: pEY + Mn · high confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Dasatinib100.00.70
Bosutinib99.20.55
Ponatinib98.50.53
Repotrectinib95.90.61
Nilotinib93.80.77
Cabozantinib91.60.75
Erdafitinib87.60.74
Tivozanib87.60.67
Ripretinib87.00.67
Crizotinib82.10.58
Fostamatinib77.30.61
Vandetanib69.40.72
Canertinib66.10.67
Afatinib35.90.71
Dacomitinib33.70.66

Known variants

No variants catalogued.
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