Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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Dasatinib

5fa423e2-ffcf-565c-8844-462f44db7406 · FDA Approved · targets BCR_ABL, ABL1, ABL2_ARG

Dasatinib

MeasuredReference

Dasatinib targets ABL2_ARG, BLK, EPHA3. Strongest hallmark effect: tumor promoting inflammation.

Top hallmarks

  • tumor promoting inflammation5.6k
  • evading apoptosis4.5k
  • proliferation4.2k

Top pathways disrupted

  • apical junction11.6k
  • allograft rejection10.9k
  • pi3k akt mtor signaling10.7k

Resistance landscape — Dasatinib

MeasuredReference

1 known oncogenic variants exist on Dasatinib's top targets — see detail for inhibition impact.

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