MP2K3
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Pralsetinib | 68.2 | 0.64 |
| Gilteritinib | 53.8 | 0.51 |
| Defactinib | 35.2 | 0.45 |
| Abemaciclib | 31.2 | 0.56 |
| Encorafenib | 29.5 | 0.76 |
| Acalabrutinib | 24.2 | 0.67 |
| Capivasertib | 18.0 | 0.64 |
| Ceritinib | 15.8 | 0.62 |
| Lenvatinib | 11.7 | 0.73 |
| Vemurafenib | 11.3 | 0.60 |
| Ibrutinib | 10.9 | 0.72 |
| Brigatinib | 10.0 | 0.51 |
| Mitapivat | 9.3 | 0.63 |
| Vandetanib | 8.4 | 0.72 |
| Remibrutinib | 8.4 | 0.72 |
Known variants
No variants catalogued.