NEK2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Neratinib | 91.1 | 0.60 |
| Infigratinib | 51.0 | 0.71 |
| Vemurafenib | 48.1 | 0.60 |
| Gilteritinib | 47.4 | 0.51 |
| Bosutinib | 46.1 | 0.55 |
| Pazopanib | 42.6 | 0.67 |
| Sunitinib | 22.0 | 0.52 |
| Tivozanib | 17.2 | 0.67 |
| Dabrafenib | 17.2 | 0.63 |
| Ripretinib | 13.7 | 0.67 |
| Fostamatinib | 13.3 | 0.61 |
| Tofacitinib | 11.4 | 0.68 |
| Dacomitinib | 11.3 | 0.66 |
| Defactinib | 10.5 | 0.45 |
| Ibrutinib | 10.3 | 0.72 |
Known variants
No variants catalogued.