Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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PAK7

RBC: PAK5 · Substrate: PAKtide ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Gilteritinib70.50.51
Brigatinib49.90.51
Pacritinib44.60.45
Defactinib43.40.45
Fostamatinib38.80.61
Capivasertib33.50.64
Sunitinib24.60.52
Pralsetinib23.60.64
Crizotinib14.90.58
Rabusertib14.20.69
Larotrectinib14.00.71
Inavolisib12.20.68
Deucravacitinib10.90.72
Capmatinib10.70.58
Midostaurin10.40.50

Known variants

No variants catalogued.
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