RPS6KA2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Brigatinib | 98.5 | 0.51 |
| Midostaurin | 98.5 | 0.50 |
| Netarsudil | 96.6 | 0.68 |
| Rabusertib | 91.1 | 0.69 |
| Sunitinib | 79.5 | 0.52 |
| Capivasertib | 71.8 | 0.64 |
| Defactinib | 67.5 | 0.45 |
| Darovasertib | 66.0 | 0.72 |
| Ceritinib | 64.7 | 0.62 |
| Bosutinib | 63.4 | 0.55 |
| Nintedanib | 57.6 | 0.61 |
| Repotrectinib | 51.5 | 0.61 |
| Lazertinib | 50.3 | 0.67 |
| Axitinib | 49.2 | 0.69 |
| Selpercatinib | 48.9 | 0.64 |
Known variants
No variants catalogued.