TGFBR2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Ponatinib | 90.8 | 0.53 |
| Vemurafenib | 86.4 | 0.60 |
| Dabrafenib | 72.6 | 0.63 |
| Pacritinib | 72.2 | 0.45 |
| Fedratinib | 41.1 | 0.58 |
| Lenvatinib | 35.5 | 0.73 |
| Erdafitinib | 32.6 | 0.74 |
| Canertinib | 30.1 | 0.67 |
| Pazopanib | 23.9 | 0.67 |
| Lorlatinib | 20.5 | 0.69 |
| Binimetinib | 19.7 | 0.69 |
| Selpercatinib | 17.2 | 0.64 |
| Gilteritinib | 17.1 | 0.51 |
| Pirtobrutinib | 17.1 | 0.66 |
| Dacomitinib | 16.4 | 0.66 |
Known variants
No variants catalogued.