TSSK2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Brigatinib | 73.9 | 0.51 |
| Ceritinib | 69.0 | 0.62 |
| Lorlatinib | 62.1 | 0.69 |
| Gilteritinib | 39.7 | 0.51 |
| Tivozanib | 31.1 | 0.67 |
| Alectinib | 26.6 | 0.65 |
| Umbralisib | 16.1 | 0.67 |
| Lazertinib | 15.8 | 0.67 |
| Defactinib | 12.8 | 0.45 |
| Selumetinib | 12.6 | 0.64 |
| Mobocertinib | 12.2 | 0.76 |
| Pacritinib | 12.1 | 0.45 |
| Infigratinib | 10.5 | 0.71 |
| Fostamatinib | 10.3 | 0.61 |
| Abrocitinib | 9.6 | 0.58 |
Known variants
No variants catalogued.