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MAP3K12(DLK/MAP3K12)

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UniProt Q12852 · PDB · AlphaFold · Substrate: MBP · Clone: Catalytic (aa 1-520)

Top inhibitors

#DrugInhibitionResidualKISSGini

Paralog block

No paralog group registered for this kinase.

EMT expression

  • Mesenchymal log2(TPM+1): 4.00
  • Epithelial log2(TPM+1): 2.71
  • Fold change: 1.29
  • Status: Upregulated

Selectivity landscape vs inhibition on MAP3K12

Each point is one of the 92 approved drugs; color = inhibition % on MAP3K12.

3D structure

Embedded NGL viewer pulls a representative PDB entry (or AlphaFold model if no experimental structure is registered). Heavy bundle — loaded only on demand.

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