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MAP3K8(COT1/MAP3K8)

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UniProt P41279 · PDB · AlphaFold · Substrate: MEK1 (K97R) · Clone: aa 30-397

Top inhibitors

#DrugInhibitionResidualKISSGini

Paralog block

No paralog group registered for this kinase.

EMT expression

  • Mesenchymal log2(TPM+1): 2.28
  • Epithelial log2(TPM+1): 2.45
  • Fold change: -0.17
  • Status: No significant change

Selectivity landscape vs inhibition on MAP3K8

Each point is one of the 92 approved drugs; color = inhibition % on MAP3K8.

3D structure

Embedded NGL viewer pulls a representative PDB entry (or AlphaFold model if no experimental structure is registered). Heavy bundle — loaded only on demand.

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