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PLK4(PLK4/SAK)

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UniProt O00444 · PDB · AlphaFold · Substrate: Casein · Clone: full-lengthmedium-confidence target

Top inhibitors

#DrugInhibitionResidualKISSGini

Paralog block

No paralog group registered for this kinase.

EMT expression

  • Mesenchymal log2(TPM+1): 3.69
  • Epithelial log2(TPM+1): 3.88
  • Fold change: -0.19
  • Status: No significant change

Selectivity landscape vs inhibition on PLK4

Each point is one of the 92 approved drugs; color = inhibition % on PLK4.

3D structure

Embedded NGL viewer pulls a representative PDB entry (or AlphaFold model if no experimental structure is registered). Heavy bundle — loaded only on demand.

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