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ROS1(ROS/ROS1)

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UniProt P08922 · PDB · AlphaFold · Substrate: IGF-1Rtide · Clone: cytoplasmic

Top inhibitors

#DrugInhibitionResidualKISSGini

Paralog block

No paralog group registered for this kinase.

EMT expression

  • Mesenchymal log2(TPM+1): 0.71
  • Epithelial log2(TPM+1): 0.07
  • Fold change: 0.63
  • Status: No significant change

Selectivity landscape vs inhibition on ROS1

Each point is one of the 92 approved drugs; color = inhibition % on ROS1.

Mutation lollipop

Cancer-associated mutations plotted by residue position. Marker size + color scale with the number of distinct cancer reports.

Variants (4)

Mutation × cancer associations

MutationCancerOrganSource
G2032Rcarcinoma_lungLungref
G2101Acarcinoma_lungLungref
G2101Ccarcinoma_lungLungref
L2086Fcarcinoma_lungLungref

3D structure

Embedded NGL viewer pulls a representative PDB entry (or AlphaFold model if no experimental structure is registered). Heavy bundle — loaded only on demand.

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