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TGFBR1(ALK5/TGFBR1)

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UniProt P36897 · PDB · AlphaFold · Substrate: Casein + Mn · Clone: aa200-503

Top inhibitors

#DrugInhibitionResidualKISSGini

Paralog block

No paralog group registered for this kinase.

EMT expression

  • Mesenchymal log2(TPM+1): 4.35
  • Epithelial log2(TPM+1): 3.23
  • Fold change: 1.12
  • Status: Upregulated

Selectivity landscape vs inhibition on TGFBR1

Each point is one of the 92 approved drugs; color = inhibition % on TGFBR1.

3D structure

Embedded NGL viewer pulls a representative PDB entry (or AlphaFold model if no experimental structure is registered). Heavy bundle — loaded only on demand.

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