b5308137-cb6a-54fa-bff3-2c01aa9a4fa2
EGFR, ERBB2_HER2
Lapatinib targets EGFR, ERBB4_HER4, ERBB2_HER2.
10 known oncogenic variants exist on Lapatinib's top targets — see detail for inhibition impact.
EGFR (A763_Y764insFHEA)
EGFR (A763_Y764insFQEA)
EGFR (A767_S768insTLA)
EGFR (C775S/T790M/L858R)
EGFR (C797A)
EGFR (C797G/L858R)
EGFR (C797S)
EGFR (C797S/L858R)
EGFR (D761Y)
EGFR (D770GY)