Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
KIRhub 2.0· v2Sign in
← Cases

EGFR

RBC: EGFR · Substrate: pEY + Mn ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Neratinib100.00.60
Mobocertinib100.00.76
Lazertinib100.00.67
Afatinib100.00.71
Gefitinib99.90.65
Dacomitinib99.80.66
Erlotinib99.40.69
Ibrutinib99.30.72
Vandetanib99.30.72
Bosutinib99.30.55
Lapatinib99.20.62
Pralsetinib99.10.64
Osimertinib99.10.73
Brigatinib98.50.51
Canertinib98.40.67

Known variants

Cancer associations

MutationCancer typeOrganSource
A750Pcarcinoma_lungLunghttps://doi.org/10.1093/nar/gkaa945
A750Plymphoid_neoplasm_haematopoietic_and_lymphoid_tissueBlood/Lymphatic Systemhttps://doi.org/10.1093/nar/gkaa945
A763carcinoma_lungLunghttps://doi.org/10.1093/nar/gkaa945
A767carcinoma_lungLunghttps://doi.org/10.1093/nar/gkaa945
A767glioma_central_nervous_systemBrain/CNShttps://doi.org/10.1093/nar/gkaa945
A767carcinoma_liverLiverhttps://doi.org/10.1093/nar/gkaa945
A767carcinoma_NSOtherhttps://doi.org/10.1093/nar/gkaa945
A767LIHCLiverhttps://doi.org/10.1093/nar/gkaa945
A767LUADLunghttps://doi.org/10.1093/nar/gkaa945
C797Gcarcinoma_lungLunghttps://doi.org/10.1093/nar/gkaa945
C797Acarcinoma_lungLunghttps://doi.org/10.1158/2159-8290.CD-12-0095
C797Scarcinoma_lungLunghttps://doi.org/10.1093/nar/gkaa945
D761Yother_lungLunghttps://doi.org/10.1093/nar/gkaa945
D761Ycarcinoma_lungLunghttps://doi.org/10.1093/nar/gkaa945
D770carcinoma_lungLunghttps://doi.org/10.1093/nar/gkaa945
D770carcinoma_endometriumUterushttps://doi.org/10.1093/nar/gkaa945
D770thymic_carcinoma_thymusThyroidhttps://doi.org/10.1093/nar/gkaa945
D770fibrous_hamartoma_of_infancy_soft_tissueSoft Tissuehttps://doi.org/10.1093/nar/gkaa945
D770carcinoma_urinary_tractBladderhttps://doi.org/10.1093/nar/gkaa945
D770glioma_central_nervous_systemBrain/CNShttps://doi.org/10.1093/nar/gkaa945
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