Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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ADRBK2

RBC: GRK3 · Substrate: Casein ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Netarsudil23.20.68
Gilteritinib18.90.51
Abrocitinib11.00.58
Ponatinib9.20.53
Ceritinib8.90.62
Fedratinib7.70.58
Asciminib7.10.60
Mobocertinib6.10.76
Tivozanib6.00.67
Brigatinib6.00.51
Capivasertib5.50.64
Crizotinib5.10.58
Sorafenib4.60.78
Pemigatinib4.60.72
Fostamatinib3.90.61

Known variants

No variants catalogued.
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