BRSK1
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Repotrectinib | 89.7 | 0.61 |
| Axitinib | 81.7 | 0.69 |
| Midostaurin | 81.4 | 0.50 |
| Brigatinib | 62.7 | 0.51 |
| Sunitinib | 43.2 | 0.52 |
| Dabrafenib | 32.2 | 0.63 |
| Defactinib | 28.2 | 0.45 |
| Rabusertib | 22.0 | 0.69 |
| Lorlatinib | 21.0 | 0.69 |
| Selpercatinib | 20.3 | 0.64 |
| Crizotinib | 14.6 | 0.58 |
| Canertinib | 13.0 | 0.67 |
| Gilteritinib | 12.4 | 0.51 |
| Nintedanib | 12.2 | 0.61 |
| Baricitinib | 10.4 | 0.62 |
Known variants
No variants catalogued.