Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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CDK15/CCNB1

RBC: CDK15/cyclin B1 · Substrate: RB Protein + Mn ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Defactinib43.70.45
Ponatinib32.80.53
Pacritinib24.20.45
Pralsetinib23.80.64
Pemigatinib23.40.72
Fedratinib14.00.58
Pexidartinib13.20.63
Repotrectinib12.40.61
Crizotinib11.50.58
Tucatinib11.30.65
Tivozanib11.20.67
Tenalisib10.60.70
Gedatolisib10.50.61
Leniolisib9.00.60
Neratinib8.90.60

Known variants

No variants catalogued.
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