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CDK6/CCND3

RBC: CDK6/cyclin D3 · Substrate: RB Protein ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Abemaciclib98.70.56
Palbociclib98.50.67
Pacritinib78.00.45
Sunitinib75.90.52
Ribociclib73.30.73
Dabrafenib66.90.63
Pemigatinib63.30.72
Defactinib49.00.45
Ponatinib45.10.53
Crizotinib36.30.58
Brigatinib27.80.51
Gilteritinib24.80.51
Fedratinib24.20.58
Trametinib23.30.72
Vemurafenib20.10.60

Known variants

No variants catalogued.
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