Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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Showing canonical CDK6/CCND1 (URL was CDK6_CYCLIN_D1).
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CDK6/CCND1

RBC: CDK6/cyclin D1 · Substrate: RB Protein ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Abemaciclib99.30.56
Palbociclib98.60.67
Ribociclib95.30.73
Pacritinib69.20.45
Defactinib56.90.45
Nintedanib51.00.61
Gilteritinib41.10.51
Sunitinib40.20.52
Brigatinib37.10.51
Vemurafenib26.90.60
Infigratinib23.70.71
Ponatinib15.30.53
Dabrafenib14.60.63
Neratinib12.60.60
Lazertinib11.20.67

Known variants

No variants catalogued.
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