CHEK1
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Rabusertib | 99.4 | 0.69 |
| Paxalisib | 95.2 | 0.61 |
| Brigatinib | 94.7 | 0.51 |
| Sunitinib | 84.2 | 0.52 |
| Nintedanib | 62.0 | 0.61 |
| Midostaurin | 60.1 | 0.50 |
| Netarsudil | 53.2 | 0.68 |
| Bosutinib | 40.7 | 0.55 |
| Gilteritinib | 30.2 | 0.51 |
| Avapritinib | 26.4 | 0.64 |
| Defactinib | 23.2 | 0.45 |
| Crizotinib | 22.5 | 0.58 |
| Capivasertib | 20.4 | 0.64 |
| Vandetanib | 19.7 | 0.72 |
| Fedratinib | 19.3 | 0.58 |
Known variants
No variants catalogued.