Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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CLK3

RBC: CLK3 · Substrate: MBP ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Bosutinib43.50.55
Ceritinib25.80.62
Dabrafenib20.50.63
Dacomitinib19.90.66
Baricitinib19.30.62
Ribociclib18.80.73
Ibrutinib18.10.72
Defactinib17.40.45
Imatinib16.00.72
Osimertinib15.40.73
Pazopanib14.40.67
Capivasertib13.70.64
Lorlatinib13.10.69
Encorafenib12.90.76
Tofacitinib12.40.68

Known variants

No variants catalogued.
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