DYRK3
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Abemaciclib | 100.0 | 0.56 |
| Defactinib | 87.7 | 0.45 |
| Palbociclib | 58.8 | 0.67 |
| Afatinib | 53.5 | 0.71 |
| Sunitinib | 47.9 | 0.52 |
| Avapritinib | 45.2 | 0.64 |
| Ponatinib | 41.2 | 0.53 |
| Gilteritinib | 40.9 | 0.51 |
| Osimertinib | 39.1 | 0.73 |
| Dacomitinib | 37.4 | 0.66 |
| Crizotinib | 36.5 | 0.58 |
| Selpercatinib | 32.6 | 0.64 |
| Neratinib | 31.7 | 0.60 |
| Gefitinib | 27.1 | 0.65 |
| Pacritinib | 25.1 | 0.45 |
Known variants
No variants catalogued.