Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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EPHA8

RBC: EPHA8 · Substrate: pEY · medium confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Bosutinib98.50.55
Dasatinib97.60.70
Ponatinib97.00.53
Nilotinib77.50.77
Vandetanib76.00.72
Ripretinib70.40.67
Repotrectinib69.90.61
Cabozantinib64.40.75
Crizotinib46.40.58
Tivozanib44.30.67
Canertinib26.30.67
Erdafitinib23.60.74
Gilteritinib21.00.51
Apatinib19.80.70
Umbralisib18.60.67

Known variants

No variants catalogued.
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