Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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HIPK1

RBC: HIPK1 · Substrate: MBP ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Abemaciclib83.60.56
Pacritinib64.30.45
Dabrafenib34.00.63
Defactinib20.40.45
Baricitinib15.10.62
Binimetinib13.90.69
Tofacitinib11.30.68
Sunitinib9.80.52
Capmatinib7.80.58
Capivasertib7.70.64
Palbociclib7.40.67
Tivozanib7.30.67
Gilteritinib5.30.51
Repotrectinib5.20.61
Abrocitinib5.10.58

Known variants

No variants catalogued.
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