IRAK4
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Vandetanib | 86.9 | 0.72 |
| Gilteritinib | 86.3 | 0.51 |
| Pacritinib | 82.8 | 0.45 |
| Sunitinib | 80.8 | 0.52 |
| Brigatinib | 76.2 | 0.51 |
| Tepotinib | 72.7 | 0.73 |
| Bosutinib | 66.4 | 0.55 |
| Alectinib | 58.1 | 0.65 |
| Defactinib | 45.7 | 0.45 |
| Midostaurin | 45.5 | 0.50 |
| Gefitinib | 42.7 | 0.65 |
| Canertinib | 33.8 | 0.67 |
| Dacomitinib | 31.8 | 0.66 |
| Pexidartinib | 30.2 | 0.63 |
| Ponatinib | 25.9 | 0.53 |
Known variants
No variants catalogued.