Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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LCK

RBC: LCK · Substrate: pEY + Mn ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Dasatinib100.00.70
Nintedanib100.00.61
Ponatinib99.70.53
Bosutinib99.70.55
Neratinib99.30.60
Vandetanib98.90.72
Repotrectinib98.60.61
Pacritinib98.40.45
Vemurafenib98.40.60
Ibrutinib98.00.72
Canertinib97.70.67
Tivozanib97.50.67
Cabozantinib97.50.75
Ripretinib97.20.67
Crizotinib96.80.58

Known variants

No variants catalogued.
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