MAP2K2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Vemurafenib | 98.1 | 0.60 |
| Bosutinib | 95.4 | 0.55 |
| Neratinib | 93.2 | 0.60 |
| Trametinib | 93.1 | 0.72 |
| Gilteritinib | 91.7 | 0.51 |
| Zanubrutinib | 89.9 | 0.79 |
| Pirtobrutinib | 89.3 | 0.66 |
| Sunitinib | 88.5 | 0.52 |
| Cabozantinib | 78.4 | 0.75 |
| Tivozanib | 74.5 | 0.67 |
| Ripretinib | 66.0 | 0.67 |
| Cobimetinib | 59.8 | 0.64 |
| Ceritinib | 53.0 | 0.62 |
| Ibrutinib | 49.2 | 0.72 |
| Canertinib | 47.3 | 0.67 |
Known variants
No variants catalogued.