Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
KIRhub 2.0· v2Sign in
← Cases

MAP2K4

RBC: MKK4 · Substrate: JNK(K55M) ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Vemurafenib58.00.60
Abemaciclib47.20.56
Defactinib38.90.45
Gilteritinib36.50.51
Osimertinib35.30.73
Pacritinib29.00.45
Midostaurin28.90.50
Pazopanib22.20.67
Ceritinib20.50.62
Capivasertib19.90.64
Sunitinib18.10.52
Dabrafenib16.90.63
Lazertinib16.80.67
Rabusertib14.30.69
Entrectinib14.30.67

Known variants

No variants catalogued.
Open in new tab