MAP3K6
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Ponatinib | 38.6 | 0.53 |
| Dabrafenib | 23.3 | 0.63 |
| Umbralisib | 19.2 | 0.67 |
| Tucatinib | 17.6 | 0.65 |
| Mitapivat | 16.2 | 0.63 |
| Selumetinib | 15.9 | 0.64 |
| Abrocitinib | 15.0 | 0.58 |
| Tepotinib | 14.4 | 0.73 |
| Avapritinib | 13.3 | 0.64 |
| Brigatinib | 13.0 | 0.51 |
| Zanubrutinib | 12.2 | 0.79 |
| Netarsudil | 11.3 | 0.68 |
| Fedratinib | 11.0 | 0.58 |
| Alpelisib | 10.7 | 0.72 |
| Bosutinib | 10.3 | 0.55 |
Known variants
No variants catalogued.