Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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MAP3K7/MAP3K7IP1

RBC: TAK1 · Substrate: Casein ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Ponatinib92.60.53
Sunitinib77.80.52
Gilteritinib76.80.51
Midostaurin74.20.50
Nintedanib67.60.61
Ripretinib52.80.67
Pacritinib43.20.45
Defactinib42.50.45
Abrocitinib34.70.58
Abemaciclib33.10.56
Sorafenib28.20.78
Bosutinib26.80.55
Regorafenib25.70.72
Dabrafenib20.30.63
Osimertinib18.70.73

Known variants

No variants catalogued.
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