Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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NTRK2

RBC: TRKB · Substrate: pEY + Mn ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Cabozantinib100.00.75
Repotrectinib99.80.61
Entrectinib99.80.67
Pralsetinib99.40.64
Alpelisib99.30.72
Crizotinib98.50.58
Ponatinib98.40.53
Larotrectinib97.90.71
Tenalisib95.30.70
Gilteritinib94.20.51
Defactinib91.30.45
Pacritinib91.20.45
Lorlatinib90.50.69
Darovasertib88.90.72
Bosutinib85.60.55

Known variants

No variants catalogued.
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