Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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PLK3

RBC: PLK3 · Substrate: Casein ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Encorafenib21.80.76
Ribociclib21.20.73
Dabrafenib19.70.63
Dacomitinib19.60.66
Ibrutinib18.50.72
Trametinib17.60.72
Tofacitinib17.10.68
Lorlatinib14.40.69
Inavolisib13.20.68
Leniolisib13.10.60
Pazopanib12.80.67
Duvelisib12.30.72
Ripretinib12.20.67
Infigratinib10.50.71
Osimertinib10.40.73

Known variants

No variants catalogued.
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