Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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ROCK1

RBC: ROCK1 · Substrate: Long S6 Kinase substrate peptide ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Netarsudil99.30.68
Capivasertib88.40.64
Baricitinib81.70.62
Ruxolitinib63.60.59
Upadacitinib47.40.66
Gilteritinib42.30.51
Abemaciclib41.90.56
Repotrectinib38.00.61
Abrocitinib29.40.58
Darovasertib25.00.72
Brigatinib24.60.51
Ceritinib22.00.62
Midostaurin21.70.50
Ponatinib21.30.53
Bosutinib17.70.55

Known variants

No variants catalogued.
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