Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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ROCK2

RBC: ROCK2 · Substrate: Long S6 Kinase substrate peptide ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Netarsudil96.00.68
Capivasertib85.60.64
Baricitinib76.50.62
Ruxolitinib49.50.59
Upadacitinib39.60.66
Abemaciclib36.60.56
Abrocitinib26.60.58
Ponatinib26.50.53
Gilteritinib24.40.51
Tivozanib22.30.67
Bosutinib20.80.55
Brigatinib14.10.51
Sunitinib13.90.52
Axitinib13.00.69
Pacritinib12.10.45

Known variants

No variants catalogued.
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