Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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RPS6KA1

RBC: RSK1 · Substrate: Glycogen Synthase-derived peptide ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Brigatinib96.10.51
Midostaurin95.50.50
Netarsudil90.10.68
Capivasertib88.80.64
Rabusertib74.30.69
Defactinib70.60.45
Sunitinib68.90.52
Ceritinib59.80.62
Nintedanib56.20.61
Gilteritinib49.10.51
Darovasertib46.30.72
Axitinib42.90.69
Alectinib40.80.65
Repotrectinib35.80.61
Selpercatinib33.60.64

Known variants

No variants catalogued.
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