Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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RPS6KA6

RBC: RSK4 · Substrate: Long S6 Kinase substrate peptide ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Midostaurin95.60.50
Brigatinib95.00.51
Sunitinib87.70.52
Defactinib84.40.45
Rabusertib84.30.69
Netarsudil83.10.68
Nintedanib69.20.61
Capivasertib66.80.64
Ceritinib56.40.62
Bosutinib53.20.55
Axitinib51.10.69
Gilteritinib50.30.51
Alectinib49.40.65
Selpercatinib47.80.64
Palbociclib40.20.67

Known variants

No variants catalogued.
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