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MAP2K1(MEK1)

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UniProt Q02750 · PDB · AlphaFold · Substrate: ERK(K52R) · Clone: full length

Top inhibitors

#DrugInhibitionResidualKISSGini
1Trametinib98.7%1.3%99.500.718
2Bosutinib89.8%10.2%87.220.555
3Pirtobrutinib81.8%18.2%99.490.656
4Cabozantinib81.2%18.8%92.730.751
5Binimetinib79.1%20.9%100.000.689
6Vemurafenib77.8%22.2%96.490.598
7Neratinib74.7%25.3%93.180.597
8Cobimetinib73.5%26.4%100.000.644
9Sunitinib68.7%31.3%91.730.524
10Tivozanib62.9%37.1%92.420.673
11Gilteritinib58.6%41.4%88.970.506
12Selumetinib54.4%45.6%100.000.640
13Zanubrutinib54.1%45.9%98.240.788
14Nintedanib46.3%53.7%90.230.608
15Capivasertib45.6%54.4%96.480.644
16Ibrutinib38.8%61.2%94.740.723
17Dasatinib34.5%65.5%87.970.699
18Abrocitinib31.8%68.2%99.500.581
19Baricitinib25.3%74.7%97.990.616
20Pacritinib19.3%80.7%88.640.452

Paralog block

No paralog group registered for this kinase.

EMT expression

  • Mesenchymal log2(TPM+1): 5.63
  • Epithelial log2(TPM+1): 5.25
  • Fold change: 0.38
  • Status: No significant change

Selectivity landscape vs inhibition on MAP2K1

Each point is one of the 92 approved drugs; color = inhibition % on MAP2K1.

Variants (1)

3D structure

Embedded NGL viewer pulls a representative PDB entry (or AlphaFold model if no experimental structure is registered). Heavy bundle — loaded only on demand.

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