Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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Erlotinib

a9f49112-77eb-597e-b033-1689b92daba5 · FDA Approved · targets EGFR

Erlotinib

MeasuredReference

Erlotinib targets EGFR, LOK_STK10, DDR1. Strongest hallmark effect: tumor promoting inflammation.

Primary targets

Top hallmarks

  • tumor promoting inflammation2.8k
  • evading apoptosis2.3k
  • proliferation2.2k

Top pathways disrupted

  • apical junction5.2k
  • pi3k akt mtor signaling4.9k
  • allograft rejection4.8k

Resistance landscape — Erlotinib

MeasuredReference

10 known oncogenic variants exist on Erlotinib's top targets — see detail for inhibition impact.

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