Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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DDR1

RBC: DDR1 · Substrate: IRS1tide · high confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Cabozantinib100.00.75
Dasatinib99.30.70
Repotrectinib99.30.61
Nilotinib98.50.77
Vandetanib98.50.72
Canertinib98.50.67
Tivozanib97.10.67
Ripretinib96.90.67
Pralsetinib96.90.64
Midostaurin96.20.50
Nintedanib96.10.61
Avapritinib96.00.64
Entrectinib96.00.67
Erdafitinib95.80.74
Gilteritinib95.70.51

Known variants

No variants catalogued.
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