Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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BLK

RBC: BLK · Substrate: pEY ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Ponatinib100.00.53
Dasatinib100.00.70
Bosutinib100.00.55
Ibrutinib99.70.72
Canertinib99.70.67
Mobocertinib99.70.76
Zanubrutinib99.10.79
Lazertinib99.00.67
Repotrectinib98.40.61
Neratinib98.20.60
Nintedanib97.60.61
Afatinib96.80.71
Pralsetinib96.10.64
Dacomitinib94.50.66
Tivozanib94.20.67

Known variants

No variants catalogued.
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