BMPR2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Defactinib | 83.5 | 0.45 |
| Deucravacitinib | 60.8 | 0.72 |
| Abemaciclib | 54.8 | 0.56 |
| Sunitinib | 52.8 | 0.52 |
| Bosutinib | 43.1 | 0.55 |
| Palbociclib | 42.3 | 0.67 |
| Gilteritinib | 41.0 | 0.51 |
| Ponatinib | 40.2 | 0.53 |
| Pacritinib | 36.3 | 0.45 |
| Alectinib | 36.2 | 0.65 |
| Avapritinib | 35.8 | 0.64 |
| Abrocitinib | 35.8 | 0.58 |
| Crizotinib | 35.6 | 0.58 |
| Selpercatinib | 34.0 | 0.64 |
| Midostaurin | 31.9 | 0.50 |
Known variants
No variants catalogued.