Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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CAMK2A

RBC: CAMK2a · Substrate: Autocamtide 2 + Ca-CaM · high confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Abemaciclib99.70.56
Brigatinib99.70.51
Alectinib97.70.65
Sunitinib96.30.52
Repotrectinib95.90.61
Ruxolitinib93.00.59
Rabusertib92.00.69
Pacritinib90.70.45
Midostaurin90.60.50
Bosutinib88.40.55
Gilteritinib81.90.51
Nintedanib80.40.61
Fedratinib68.00.58
Baricitinib62.80.62
Palbociclib53.70.67

Known variants

No variants catalogued.
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