Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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CAMK2G

RBC: CAMK2g · Substrate: ZIPtide + Ca-CaM* ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Brigatinib92.70.51
Abemaciclib82.00.56
Alectinib58.60.65
Sunitinib49.00.52
Midostaurin33.20.50
Crizotinib32.80.58
Ruxolitinib28.80.59
Rabusertib22.90.69
Pacritinib20.40.45
Dabrafenib19.30.63
Ponatinib18.90.53
Repotrectinib17.20.61
Encorafenib16.30.76
Tofacitinib16.20.68
Ibrutinib15.30.72

Known variants

No variants catalogued.
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