CHEK2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Brigatinib | 99.4 | 0.51 |
| Alectinib | 98.8 | 0.65 |
| Sunitinib | 95.0 | 0.52 |
| Ponatinib | 92.6 | 0.53 |
| Bosutinib | 91.4 | 0.55 |
| Ceritinib | 88.8 | 0.62 |
| Selpercatinib | 86.3 | 0.64 |
| Netarsudil | 86.0 | 0.68 |
| Gilteritinib | 82.5 | 0.51 |
| Neratinib | 76.1 | 0.60 |
| Vandetanib | 58.3 | 0.72 |
| Fedratinib | 50.0 | 0.58 |
| Cabozantinib | 43.3 | 0.75 |
| Defactinib | 38.9 | 0.45 |
| Lazertinib | 35.3 | 0.67 |