DCLK1
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Lorlatinib | 77.5 | 0.69 |
| Crizotinib | 69.0 | 0.58 |
| Ceritinib | 65.2 | 0.62 |
| Baricitinib | 64.7 | 0.62 |
| Brigatinib | 58.4 | 0.51 |
| Ruxolitinib | 39.3 | 0.59 |
| Fedratinib | 36.5 | 0.58 |
| Dabrafenib | 25.4 | 0.63 |
| Sunitinib | 23.3 | 0.52 |
| Palbociclib | 18.5 | 0.67 |
| Abemaciclib | 17.9 | 0.56 |
| Pemigatinib | 17.6 | 0.72 |
| Gilteritinib | 15.4 | 0.51 |
| Entrectinib | 13.9 | 0.67 |
| Defactinib | 10.8 | 0.45 |
Known variants
No variants catalogued.