Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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DMPK

RBC: DMPK · Substrate: SGKtide ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Darovasertib27.30.72
Bosutinib24.00.55
Fostamatinib10.30.61
Trametinib10.20.72
Imatinib10.00.72
Ribociclib8.70.73
Nintedanib8.10.61
Baricitinib8.10.62
Ponatinib8.00.53
Everolimus7.50.71
Ruxolitinib7.20.59
Crizotinib7.10.58
Vemurafenib6.60.60
Entrectinib6.50.67
Dacomitinib6.40.66

Known variants

No variants catalogued.
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