DYRK2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Abemaciclib | 97.1 | 0.56 |
| Selpercatinib | 75.9 | 0.64 |
| Defactinib | 74.8 | 0.45 |
| Afatinib | 62.6 | 0.71 |
| Osimertinib | 62.1 | 0.73 |
| Palbociclib | 53.2 | 0.67 |
| Dacomitinib | 52.1 | 0.66 |
| Ponatinib | 51.5 | 0.53 |
| Pacritinib | 46.0 | 0.45 |
| Sunitinib | 37.2 | 0.52 |
| Avapritinib | 36.8 | 0.64 |
| Crizotinib | 35.9 | 0.58 |
| Midostaurin | 35.6 | 0.50 |
| Brigatinib | 34.4 | 0.51 |
| Erlotinib | 29.6 | 0.69 |
Known variants
No variants catalogued.